Arylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties

Baranovskyi, Vitaliy; Symchak, Ruslan; Pokryshko, Olena; Klymnyuk, Sergiy; Grishchuk, Bogdan

Please use this identifier to cite or link to this item: https://oldena.lpnu.ua/handle/ntb/45209

Title:	Arylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties
Other Titles:	Арилзаміщені галогено(тіоціанато)аміди, що містять 4-ацетилфенільний фрагмент. Синтез, циклізація та протимікробні властивості
Authors:	Baranovskyi, Vitaliy Symchak, Ruslan Pokryshko, Olena Klymnyuk, Sergiy Grishchuk, Bogdan
Affiliation:	Ternopil V. Hnatyuk National Pedagogical University I. Ya. Horbachevsky Ternopil State Medical University
Bibliographic description (Ukraine):	Arylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties / Vitaliy Baranovskyi, Ruslan Symchak, Olena Pokryshko, Sergiy Klymnyuk, Bogdan Grishchuk // Chemistry & Chemical Technology. — Lviv : Lviv Politechnic Publishing House, 2018. — Vol 12. — No 4. — P. 447–450.
Bibliographic description (International):	Arylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties / Vitaliy Baranovskyi, Ruslan Symchak, Olena Pokryshko, Sergiy Klymnyuk, Bogdan Grishchuk // Chemistry & Chemical Technology. — Lviv : Lviv Politechnic Publishing House, 2018. — Vol 12. — No 4. — P. 447–450.
Is part of:	Chemistry & Chemical Technology, 4 (12), 2018
Journal/Collection:	Chemistry & Chemical Technology
Issue:	4
Volume:	12
Issue Date:	20-Jan-2018
Publisher:	Lviv Politechnic Publishing House
Place of the edition/event:	Lviv
Keywords:	аніонарилювання аміди акрилової і метакрилової кислот солі 4-ацетилфенілдіазонію 5-арилза- міщені 2-амінотіазол-4(5Н)-они протимікробна активність anionarylation acrylic and methacrylic acids amides 4-acetylphenyldiazonium salts 5-arylsubstituted 2-aminothiazol-4(5H)-ones antimicrobial activity
Number of pages:	4
Page range:	447-450
Start page:	447
End page:	450
Abstract:	Купрокаталітичним аніонарилюванням амідів акрилової і метакрилової кислот солями 4-ацетилфе- нілдіазонію синтезовані 3-(4-ацетилфеніл)-(2-метил)-2-хлоро (бромо, тіоціанато)пропанаміди. Циклізацією тіоціанато- амідів одержані арилзаміщені 2-амінотіазол-4(5Н)-они з ацетофеноновим фрагментом. Досліджено протибакте- ріальну та протигрибкову активність синтезованих сполук. 13-(4-Acetylphenyl)-(2-methyl)-2-chloro(bromo, thiocyanato)propanamides have been obtained via copper catalytic anionarylation of acrylic and methacrylic acids amides by 4-acetylphenyldiazonium salts. 5-(4-Acetylphenyl) substituted 2-aminothiazol-4(5H)-ones were synthesized by cyclisation of thiocyanatoamides. All synthesized compounds were tested for their antibacterial and antomycotic activity.
URI:	https://ena.lpnu.ua/handle/ntb/45209
Copyright owner:	© Національний університет „Львівська політехніка“, 2018 ©Baranovskyi V., Symchak R., Pokryshko O., Klymnyuk S.,Grishchuk B., 2018
URL for reference material:	https://doi.org/10.1042/bj1520233 https://doi.org/10.3390/molecules15128813 https://doi.org/10.1039/C5MD00357A https://doi.org/10.1134/S1070363209020170 https://doi.org/10.1134/S1070363214080106 https://doi.org/10.1007/s11094-011-0673-0 https://doi.org/10.1007/s11094-013-0949-7 https://doi.org/10.1007/s11094-016-1484-0 https://doi.org/10.23939/chcht09.02.193
References (Ukraine):	[1] O'Neil M. (Ed.): The Merck Index: An Encyclopedia of Chemicals, Drugs, and Biologicals, 15th edn. Merck and Co. Inc., Cambridge 2013. [2] Cripps R.: Biochem J., 1975, 152, 233.https://doi.org/10.1042/bj1520233 [3] Salas P., Soto A., Carretero A. et al.:Molecules, 2010, 15,8813. https://doi.org/10.3390/molecules15128813 [4] Pharmaceutical Manufacturing Encyclopedia. William Andrew Publishing, Norwich, NY 2007. [5] Shen Y., Li B., Xu H. et al.: Pharmazie, 2013, 68, 307. [6] Wang Z., Li X., Xu W. et al.:Med. Chem. Commun., 2015, 6,2146. https://doi.org/10.1039/C5MD00357A [7] Baranovskii V., Simchak R., Grishchuk B.: Russ. J. Gen. Chem.,2009, 79, 269. https://doi.org/10.1134/S1070363209020170 [8] Baranovskii V., Yatsyuk V., Grishchuk B.: Russ. J. Gen. Chem.,2014, 84, 1505. https://doi.org/10.1134/S1070363214080106 [9] Grishchuk B., Baranovskii V., Klymnyuk S. et al.: Pharm. Chem. J., 2011, 45, 532. https://doi.org/10.1007/s11094-011-0673-0 [10] Grishchuk B., Simchak R., Baranovskii V. et al.: Pharm. Chem. J., 2013, 47, 307. https://doi.org/10.1007/s11094-013-0949-7 [11] Grishchuk B., Yatsyuk V., Baranovskii V. et al.: Pharm. Chem. J., 2016, 50, 534. https://doi.org/10.1007/s11094-016-1484-0 [12] Yatsyuk V., Pokryshko O., Yaniv Z. et al.: Chem. Chem. Technol., 2015, 9, 193. https://doi.org/10.23939/chcht09.02.193 [13] Grishchuk B., Baranovskyi V., Klymnyuk S.: Pharmac. Rev.,2011, 4, 117.
References (International):	[1] O'Neil M. (Ed.): The Merck Index: An Encyclopedia of Chemicals, Drugs, and Biologicals, 15th edn. Merck and Co. Inc., Cambridge 2013. [2] Cripps R., Biochem J., 1975, 152, 233.https://doi.org/10.1042/bj1520233 [3] Salas P., Soto A., Carretero A. et al.:Molecules, 2010, 15,8813. https://doi.org/10.3390/molecules15128813 [4] Pharmaceutical Manufacturing Encyclopedia. William Andrew Publishing, Norwich, NY 2007. [5] Shen Y., Li B., Xu H. et al., Pharmazie, 2013, 68, 307. [6] Wang Z., Li X., Xu W. et al.:Med. Chem. Commun., 2015, 6,2146. https://doi.org/10.1039/P.5MD00357A [7] Baranovskii V., Simchak R., Grishchuk B., Russ. J. Gen. Chem.,2009, 79, 269. https://doi.org/10.1134/S1070363209020170 [8] Baranovskii V., Yatsyuk V., Grishchuk B., Russ. J. Gen. Chem.,2014, 84, 1505. https://doi.org/10.1134/S1070363214080106 [9] Grishchuk B., Baranovskii V., Klymnyuk S. et al., Pharm. Chem. J., 2011, 45, 532. https://doi.org/10.1007/s11094-011-0673-0 [10] Grishchuk B., Simchak R., Baranovskii V. et al., Pharm. Chem. J., 2013, 47, 307. https://doi.org/10.1007/s11094-013-0949-7 [11] Grishchuk B., Yatsyuk V., Baranovskii V. et al., Pharm. Chem. J., 2016, 50, 534. https://doi.org/10.1007/s11094-016-1484-0 [12] Yatsyuk V., Pokryshko O., Yaniv Z. et al., Chem. Chem. Technol., 2015, 9, 193. https://doi.org/10.23939/chcht09.02.193 [13] Grishchuk B., Baranovskyi V., Klymnyuk S., Pharmac. Rev.,2011, 4, 117.
Content type:	Article
Appears in Collections:	Chemistry & Chemical Technology. – 2018. – Vol. 12, No. 4

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